Multiparametric Assays for Accelerating Early Drug Discovery: Trends in Pharmacological Sciences
Drug Target Identification Methods After a Phenotypic Screen - Drug Hunter
Target Engagement Studies with Syngeneic Tumor Models
Target Engagement Measures in Preclinical Drug Discovery: Theory, Methods, and Case Studies | SpringerLink
CETSA: a target engagement assay with potential to transform drug discovery. | Semantic Scholar
Target Engagement in Lead Generation - ScienceDirect
Kinase Biology for Drug Discovery
Promega Launches NanoBRET™ Target Engagement Intracellular Kinase Assay, First to Quantitatively Measure Drug-Kinase Interactions in Live Cells | Business Wire
Monitoring Target Engagement In Drug Discovery Application Of Wes To The Cellular Thermal Shift Assay
CETSA: a target engagement assay with potential to transform drug discovery | Future Medicinal Chemistry
Cellular Thermal Shift Assays - bringing relevant target engagement to your drug discovery workflow - Drug Target Review
Target engagement approaches for pharmacological evaluation in animal models - Chemical Communications (RSC Publishing)
NanoBRET Target Engagement | Live-Cell Compound Binding Assay
Frontiers | Current Advances in CETSA
Target engagement and drug residence time can be observed in living cells with BRET | Nature Communications
Promega NanoLuc Enables a First in Measuring Drug-Target Residence in Live Cells | Business Wire
Mass spectrometry-based Cellular Thermal Shift Assay (CETSA®) for target deconvolution in phenotypic drug discovery - ScienceDirect
Sensitive Measurement of Drug-Target Engagement by a Cellular Thermal Shift Assay with Multiplex Proximity Extension Readout | Analytical Chemistry
Biomarkers in efficacy and safety assessments. Application of in vitro... | Download Scientific Diagram
DNA-Encoded Libraries (DELs) and NanoBRET™ Target Engagement Assays Accelerate Drug Discovery
Alpha CETSA Human Cereblon Target Engagement Detection Kit, Lysis Buffer 4, 5,000 Assay Points | PerkinElmer
Determining target engagement in living systems | Nature Chemical Biology
Assessing target engagement using proteome-wide solvent shift assays | eLife
Target Engagement in Lead Generation - ScienceDirect
Target Engagement Reagents | PerkinElmer
